yana-notes

Methylphenylpiracetam

2025-02-08:

MethylPhenylpiracetam #

σ1 PAM.

  • 211% memory boost in mice models, no toxicity noticed in mice, rat, or monkey models, no tolerance build up
  • E1R is the erythro- enantiomer, which has the greatest effect.
Enantiomer σ1R PAM effect %
erythro-(4R,5S) 222 ± 37
threo-(4R,5R) 191 ± 23
erythro-(4S,5R) 141 ± 40
threo-(4S,5S) 147 ± 31