yana-notes

GTS-21

2022-03-02: Drugs reference:

GTS-21 (DXMBA) 150 #

Partial agonist of α7 nAChR. Technically binds to α4β2 nAChR antagonizing it, but insignificant activation.

  • Had no effect on locomotor activity in mice or dopamine turnover in rats. R

Supplementation #

1.7 hour half life and really expensive.