yana-notes

Pramipexole

2022-07-05: reference:

Pramipexole #

Treats Parkinson’s and restless leg syndrome.

Site Affinity (Ki, nM) Efficacy (Emax, %) Action
D2S 3.9 130 Full agonist
D2L 2.2 70 Partial agonist
D3 0.5 70 Partial agonist
D4 5.1 42 Partial agonist