yana-notes

Acetylcholinesterase

links: reference: 10-18-2021

Acetylcholinesterase (AChE) #

  • Don’t forget about the other cholinesterase, butyrylcholinesterase (synthetic). Dual cholinesterase inhibitors work on both of these.
  • Non-fearful rats have a ton of this stuff, and AChE-KO mice have increased Depression an anxiety-like behavior.

Inhibitors #

  • So I think they differ a lot - especially with herbals, which usually produce AChEis as a toxic defense mechanism. They could have different binding affinities for certain regions, which is obviously pretty relevant.
  • Inhibitors cause Gyno through unknown mechanisms.
  • Scopolamine and datura are pretty potent AChE inhibitors, raising ACh levels in the brain, but their strong antimuscarinic properties far overshadows this.